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IRIS è il sistema di gestione integrata dei dati della ricerca (persone, progetti, pubblicazioni, attività) adottato dall'Università degli Studi di Cagliari dal mese di luglio 2015.

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TitoloData di pubblicazioneAutore(i)RivistaEditore
Targeting tumor associated carbonic anhydrase IX and XII: Highly isozyme selective coumarin and psoralen inhibitors2018Melis, Claudia; Distinto, Simona; Bianco, Giulia; Meleddu, Rita; Cottiglia, Filippo; Fois, Benede...tta; Taverna, Domenico; Angius, Rossella; Alcaro, Stefano; Ortuso, Francesco; Gaspari, Marco; Angeli, Andrea; Del Prete, Sonia; Capasso, Clemente; Supuran, Claudiu T.; Maccioni, EliasACS MEDICINAL CHEMISTRY LETTERS
Tuning the Dual Inhibition of Carbonic Anhydrase and Cyclooxygenase by Dihydrothiazole Benzensulfonamides2018Meleddu, Rita; Distinto, Simona; Cottiglia, Filippo; Angius, Rossella; Gaspari, Marco; Taverna, D...omenico; Melis, Claudia; Angeli, Andrea; Bianco, Giulia; Deplano, Serenella; Fois, Benedetta; Del Prete, Sonia; Capasso, Clemente; Alcaro, Stefano; Ortuso, Francesco; Yanez, Matilde; Supuran Claudiu, T.; Maccioni, EliasACS MEDICINAL CHEMISTRY LETTERS
Identification of Myricetin as Ebolavirus VP35-dsRNA interaction inhibitor through a novel fluorescence-based assay2018Luca Daino, Gian; Frau, Aldo; Sanna, Cinzia; Rigano, Daniela; Distinto, Simona; Madau, Veronica; ...Esposito, Francesca; Fanunza, Elisa; Bianco, Giulia; Taglialatela-Scafati, Orazio; Zinzula, Luca; Maccioni, Elias; Corona, Angela; Tramontano, EnzoBIOCHEMISTRY
Through scaffold modification to 3,5-diaryl-4,5-dihydroisoxazoles: new potent and selective inhibitors of monoamine oxidase B2017Meleddu, Rita; Distinto, Simona; Cirilli, Roberto; Alcaro, Stefano; Yanez, Matilde; Sanna, Maria ...Luisa; Corona, Angela; Melis, Claudia; Bianco, Giulia; Matyus, Peter; Cottiglia, Filippo; Maccioni, EliasJOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
Design, synthesis and antiviral evaluation of novel heteroarylcarbothioamide derivatives as dual inhibitors of HIV-1 Reverse transcriptase-associated RNase H and RDDP functions2017Corona, Angela; Onnis, Valentina; Deplano, Alessandro; Bianco, Giulia; Demurtas, Monica; Distinto..., Simona; Cheng, Yung Chi; Alcaro, Stefano; Esposito, Francesca; Tramontano, EnzoPATHOGENS AND DISEASE
Phenylpropenoids from Bupleurum fruticosum as Anti-Human Rhinovirus Species A Selective Capsid Binders2017Fois, Benedetta; Bianco, Giulia; Sonar, Vijay P.; Distinto, Simona; Maccioni, Elias; Meleddu, Rit...a; Melis, Claudia; Marras, Luisa; Pompei, Raffaello; Floris, Costantino; Caboni, Pierluigi; Cottiglia, FilippoJOURNAL OF NATURAL PRODUCTS
N-Acylbenzenesulfonamide dihydro-1,3,4-oxadiazole hybrids: seeking selectivity toward carbonic anhydrase isoforms2017Bianco, Giulia; Meleddu, Rita; Distinto, Simona; Cottiglia, Filippo; Gaspari, Marco; Melis, Claud...ia; Corona, Angela; Angius, Rossella; Angeli, Andrea; Taverna, Domenico; Alcaro, Stefano; Leitans, Janis; Kazaks, Andris; Tars, Kaspars; Supuran, Claudiu T.; Maccioni, EliasACS MEDICINAL CHEMISTRY LETTERS
Isatin thiazoline hybrids as dual inhibitors of HIV-1 reverse transcriptase2017Meleddu, Rita; Distinto, Simona; Corona, Angela; Tramontano, Enzo; Bianco, Giulia; Melis, Claudia...; Cottiglia, Filippo; Maccioni, EliasJOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
Isatin: a privileged scaffold for the design of carbonic anhydrase inhibitors2017Melis, Claudia; Meleddu, Rita; Angeli, Andrea; Distinto, Simona; Bianco, Giulia; Capasso, Clement...e; Cottiglia, Filippo; Angius, Rossella; Supuran, Claudiu T.; Maccioni, EliasJOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
Structure-based approaches applied to the study of pharmaceutical relevant targets24-mar-2016Università degli Studi di Cagliari
Exploring the thiazole scaffold for the identification of new agents for the treatment of fluconazole resistant Candida2016Meleddu, Rita; Distinto, Simona; Corona, Angela; Maccioni, Elias; Arridu, Antonella; Melis, Claud...ia; Bianco, Giulia; Matyus, Peter; Cottiglia, Filippo; Sanna, Adriana; DE LOGU, AlessandroJOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
Drug design, synthesis, in vitro and in silico evaluation of selective monoaminoxidase B inhibitors based on 3-acetyl-2-dichlorophenyl-5-aryl-2,3-dihydro-1,3,4-oxadiazole chemical scaffold2016Distinto, Simona; Meleddu, Rita; Yanez, Matilde; Cirilli, Roberto; Bianco, Giulia; Sanna, Maria L...uisa; Arridu, Antonella; Cossu, Pietro; Cottiglia, Filippo; Faggi, Cristina; Ortuso, Francesco; Alcaro, Stefano; Maccioni, EliasEUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
Ribonuclease H/DNA polymerase HIV-1 reverse transcriptase dual inhibitor: mechanistic studies on the allosteric mode of action of isatin-based compound RMNC62016Corona, A; Meleddu, R; Esposito, F; Distinto, S; Bianco, G; Masaoka, T; Maccioni, E; Menéndez-Ari...as, L; Alcaro, S; Le Grice, SFJ; Tramontano, EPLOS ONE
(3Z)-3-(2-[4-(aryl)-1,3-thiazol-2-yl]hydrazin-1-ylidene)-2,3-dihydro- 1H -indol-2-one derivatives as dual inhibitors of HIV-1 reverse transcriptase2015Meleddu, Rita; Distinto, Simona; Corona, Angela; Bianco, Giulia; Cannas, Valeria; Esposito, Franc...esca; Artese, A; Alcaro, S; Matyus, P; Bogdan, D; Cottiglia, Filippo; Tramontano, Enzo; Maccioni, EliasEUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
New 4-[(3-cyclohexyl-4-aryl-2,3-dihydro-1,3-thiazol-2-ylidene)amino]benzene-1-sulfonamides, synthesis and inhibitory activity toward carbonic anhydrase I, II, IX, XII2015Meleddu, Rita; Maccioni, Elias; Distinto, Simona; Bianco, Giulia; Melis, Claudia; Alcaro, Stefano...; Cottiglia, Filippo; Ceruso, Mariangela; Supuran, Claudiu T.BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
Design, synthesis and biological activity evaluation of c-myc proto-oncogene binders as potential antitumor agents2013Meleddu, R.; Distinto, S; Sissi, C.; Musetti, C.; Arridu, A.; Bianco, Giulia; Parrotta, L.; Ortus...o, F.; Alcaro, S.; Maccioni, Elias
2-(2-cycloalkylidene hydrazin-1-yl)-4-aryl-1,3-thiazoles: a promising class of antifungal agents2013Arridu A.; Meleddu R.; Bianco G.; Distinto S.; De Logu A.; Matyus P.; Maccioni E
Towards the total block of HIV-1 Reverse Transcriptase: the dual-inhibitors approach2013Meleddu R.; Arridu A.; Bianco G.; Tramontano E.; Distinto S.; Matyus P.; Maccioni E
In search of new antitumor agents through the combination of individually active moieties: construction of a [3,5-diaryl-(4,5- dihydropyrazol-1-yl)-4-oxo-1,3-thiazol-5-ylidene]- 1H-indol-2-ones library2013Arridu A.; Meleddu R.; Bianco G; Distinto S; Bogdan D.; Matyus P.; Maccioni E.
MD protocol validation for the study of MAOB-inhibitor complexes2013Bianco G.; Cossu P.; Distinto S.; Meleddu R.; Arridu A.; Ortuso F.; Alcaro S.; Maccioni E
   
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