Titolo | Data di pubblicazione | Autori | Tipo | Abstract |
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Dual HIV-1 reverse transcriptase and integrase inhibitors from Limonium morisianum Arrigoni, an endemic species of Sardinia (Italy) | 2019 | SANNA, CINZIA ; Daniela, Rigano; CORONA, ANGELA ; PIANO, DARIO ; Carmen, Formisano; FARCI, DOMENICA ; Genni, Franzini; BALLERO, MAURO ; Giuseppina, Chianese; TRAMONTANO, ENZO ; Orazio, Taglialatela-Scafati; ESPOSITO, FRANCESCA | 1 Contributo su Rivista::1.1 Articolo in rivista | |
Chromenone derivatives as a versatile scaffold with dual mode of inhibition of HIV-1 reverse transcriptase-associated Ribonuclease H function and integrase activity | 2019 | ESPOSITO, FRANCESCA ; Ambrosio F. A.; Maleddu R.; Costa G.; Rocca R.; MACCIONI, ELIAS ; Catalano R.; Romeo I.; Eleftheriou P.; Karia D. C.; Tsirides P.; Godvani N.; Pandya H.; Alcaro S.; Artese A.; GERONIKAKI, ATHINA ; TRAMONTANO, ENZO | 1 Contributo su Rivista::1.1 Articolo in rivista | |
Prenylated phloroglucinols from Hypericum scruglii, an endemic species of Sardinia (Italy), as new dual HIV-1 inhibitors effective on HIV-1 replication | 2018 | SANNA, CINZIA ; Monica Scognamiglio; Antonio Fiorentino; CORONA, ANGELA ; Vittoria Graziani; CAREDDA, ALESSIA ; CORTIS, PIERLUIGI ; Mariofilippo Montisci; Elisa Rita Ceresola; Filippo Canducci; Ferruccio Poli; TRAMONTANO, ENZO ; ESPOSITO, FRANCESCA | 1 Contributo su Rivista::1.1 Articolo in rivista | |
Identification of Myricetin as Ebolavirus VP35-dsRNA interaction inhibitor through a novel fluorescence-based assay | 2018 | Gian Luca Daino; FRAU, ALDO ; SANNA, CINZIA ; Daniela Rigano; DISTINTO, SIMONA ; MADAU, VERONICA ; ESPOSITO, FRANCESCA ; FANUNZA, ELISA ; BIANCO, GIULIA ; Orazio Taglialatela-Scafati; ZINZULA, LUCA ; MACCIONI, ELIAS ; CORONA, ANGELA ; TRAMONTANO, ENZO | 1 Contributo su Rivista::1.1 Articolo in rivista | |
Improvement of the activity of the anti-HIV-1 integrase aptamer T30175 by introducing a modified thymidine into the loops | 2018 | Virgilio, Antonella; Amato, Teresa; Petraccone, Luigi; ESPOSITO, FRANCESCA ; GRANDI, NICOLE ; TRAMONTANO, ENZO ; Romero, Raquel; Haider, Shozeb; Gomez-Monterrey, Isabel; Novellino, Ettore; Mayol, Luciano; Esposito, Veronica; Galeone, Aldo | 1 Contributo su Rivista::1.1 Articolo in rivista | |
Structure-guided approach identifies a novel class of HIV-1 Ribonuclease H inhibitors: Binding mode insights through magnesium complexation and site-directed mutagenesis studies | 2018 | Vasanthanathan Poongavanam; CORONA, ANGELA ; Casper Svendsen; Luigi Scipione; GRANDI, NICOLE ; Fabiana Pandolfi; Roberto Di Santo; Roberta Costi; ESPOSITO, FRANCESCA ; TRAMONTANO, ENZO ; Jacob Kongsted | 1 Contributo su Rivista::1.1 Articolo in rivista | |
Onopordum illyricum L., a Mediterranean plant, as a source of anti HIV-1 compounds | 2018 | SANNA, CINZIA ; D. Rigano; CORTIS, PIERLUIGI ; CORONA, ANGELA ; BALLERO, MAURO ; C. Parolin; C. Del Vecchio; G. Chianese; E. Saccon; C. Formisano; TRAMONTANO, ENZO ; ESPOSITO, FRANCESCA | 1 Contributo su Rivista::1.1 Articolo in rivista | |
On the S-layer of Thermus thermophilus and the assembling of its main protein SIpA | 2018 | FARCI, DOMENICA ; Farci, Stefano Francesco; ESPOSITO, FRANCESCA ; TRAMONTANO, ENZO ; Kirkpatrick, Joanna; PIANO, DARIO | 1 Contributo su Rivista::1.1 Articolo in rivista | |
Identification of a novel HERV-K(HML10): comprehensive characterization and comparative analysis in non-human primates provide insights about HML10 proviruses structure and diffusion | 2017 | GRANDI, NICOLE ; CADEDDU, MARTA ; PISANO, MARIA PAOLA ; ESPOSITO, FRANCESCA ; Blomberg, Jonas; TRAMONTANO, ENZO | 1 Contributo su Rivista::1.1 Articolo in rivista | |
Design, synthesis and antiviral evaluation of novel heteroarylcarbothioamide derivatives as dual inhibitors of HIV-1 Reverse transcriptase-associated RNase H and RDDP functions | 2017 | CORONA, ANGELA ; ONNIS, VALENTINA ; DEPLANO, ALESSANDRO ; BIANCO, GIULIA ; DEMURTAS, MONICA ; DISTINTO, SIMONA ; Cheng, Yung Chi; Alcaro, Stefano; ESPOSITO, FRANCESCA ; TRAMONTANO, ENZO | 1 Contributo su Rivista::1.1 Articolo in rivista | |
Natural Product Kuwanon-L Inhibits HIV-1 Replication through Multiple Target Binding | 2017 | Martini, Riccardo; ESPOSITO, FRANCESCA ; CORONA, ANGELA ; Ferrarese, Roberto; Ceresola, Elisa Rita; Visconti, Laura; Tintori, Cristina; Barbieri, Alessandro; Calcaterra, Andrea; Iovine, Valentina; Canducci, Filippo; TRAMONTANO, ENZO ; Botta, Maurizio | 1 Contributo su Rivista::1.1 Articolo in rivista | |
Chelation motifs affecting metal-dependent viral enzymes: N′-acylhydrazone ligands as dual target inhibitors of HIV-1 Integrase and Reverse Transcriptase Ribonuclease H domain | 2017 | Carcelli, Mauro; Rogolino, Dominga; Gatti, Anna; Pala, Nicolino; CORONA, ANGELA ; CAREDDA, ALESSIA ; TRAMONTANO, ENZO ; Pannecouque, Christophe; Naesens, Lieve; ESPOSITO, FRANCESCA | 1 Contributo su Rivista::1.1 Articolo in rivista | |
Multi-target activity of Hemidesmus indicus decoction against innovative HIV-1 drug targets and characterization of Lupeol mode of action | 2017 | ESPOSITO, FRANCESCA ; Mandrone, Manuela; Del Vecchio, Claudia; Carli, Ilaria; DISTINTO, SIMONA ; CORONA, ANGELA ; Lianza, Mariacaterina; PIANO, DARIO ; Tacchini, Massimo; MACCIONI, ELIAS ; COTTIGLIA, FILIPPO ; Saccon, Elisa; Poli, Ferruccio; Parolin, Cristina; TRAMONTANO, ENZO | 1 Contributo su Rivista::1.1 Articolo in rivista | |
S-layer proteins as a source of carotenoids: Isolation of the carotenoid cofactor deinoxanthin from its S-layer protein DR_2577 | 2017 | FARCI, DOMENICA ; ESPOSITO, FRANCESCA ; El Alaoui, Sabah; PIANO, DARIO | 1 Contributo su Rivista::1.1 Articolo in rivista | |
New insights into the operative network of FaEO, an enone oxidoreductase from Fragaria x ananassa Duch | 2017 | COLLU, GABRIELLA ; FARCI, DOMENICA; ESPOSITO, FRANCESCA ; PINTUS, FRANCESCA ; Kirkpatrick, Joanna; PIANO, DARIO | 1 Contributo su Rivista::1.1 Articolo in rivista | |
New insights into the interaction between pyrrolyl diketoacids and HIV-1 integrase active site and comparison with RNase H | 2016 | CORONA, ANGELA ; di Leva, Francesco Saverio; Rigogliuso, Giuseppe; Pescatori, Luca; Madia, Valentina Noemi; Subra, Frederic; Delelis, Olivier; ESPOSITO, FRANCESCA ; CADEDDU, MARTA ; Costi, Roberta; Cosconati, Sandro; Novellino, Ettore; di Santo, Roberto; TRAMONTANO, ENZO | 1 Contributo su Rivista::1.1 Articolo in rivista | |
Studies on Cycloheptathiophene-3-carboxamide Derivatives as Allosteric HIV-1 Ribonuclease H Inhibitors | 2016 | CORONA, ANGELA ; Desantis, Jenny; Massari, Serena; DISTINTO, SIMONA ; Masaoka, Takashi; Sabatini, Stefano; ESPOSITO, FRANCESCA ; Manfroni, Giuseppe; MACCIONI, ELIAS ; Cecchetti, Violetta; Pannecouque, Christophe; Le Grice, Stuart F. J; TRAMONTANO, ENZO ; Tabarrini, Oriana | 1 Contributo su Rivista::1.1 Articolo in rivista | |
Inhibition of HIV-1 reverse transcriptase dimerization by small molecules | 2016 | Tintori, C; CORONA, ANGELA ; ESPOSITO, FRANCESCA ; Brai, A; GRANDI, NICOLE ; Ceresola, ER; Clementi, M; Canducci, F; TRAMONTANO, ENZO ; Botta, M. | 1 Contributo su Rivista::1.1 Articolo in rivista | |
Ribonuclease H/DNA polymerase HIV-1 reverse transcriptase dual inhibitor: mechanistic studies on the allosteric mode of action of isatin-based compound RMNC6 | 2016 | CORONA, ANGELA ; MELEDDU, RITA ; ESPOSITO, FRANCESCA ; DISTINTO, SIMONA ; BIANCO, GIULIA ; Masaoka, T; MACCIONI, ELIAS ; Menéndez Arias, L; Alcaro, S; Le Grice, SFJ; TRAMONTANO, ENZO | 1 Contributo su Rivista::1.1 Articolo in rivista | |
Development and identification of a novel anti-HIV-1 peptide derived by modification of the N-terminal domain of HIV-1 integrase | 2016 | Sala, M; Spensiero, A; ESPOSITO, FRANCESCA ; Scala, MC; Vernieri, E; Bertamino, A; Manfra, M; Carotenuto, A; Grieco, P; Novellino, E; CADEDDU, MARTA ; TRAMONTANO, ENZO ; Schols, D; Campiglia, P; Gomez Monterrey, IM | 1 Contributo su Rivista::1.1 Articolo in rivista | |