{"id":45,"date":"2009-12-02T01:05:59","date_gmt":"2009-12-01T23:05:59","guid":{"rendered":"http:\/\/people.unica.it\/ivconvegnonpcf\/?page_id=45"},"modified":"2010-05-03T20:55:09","modified_gmt":"2010-05-03T18:55:09","slug":"programma-scientifico","status":"publish","type":"page","link":"https:\/\/people.unica.it\/ivconvegnonpcf\/il-congresso\/programma-scientifico\/","title":{"rendered":"Programma del Convegno"},"content":{"rendered":"

\u00a0IV Meeting \u201cNuove Prospettive in Chimica Farmaceutica\u201d<\/span><\/em><\/strong><\/p>\n

\u00a0<\/strong><\/span><\/p>\n

Gioved\u00ec 06\/05\/2010<\/span><\/strong><\/span><\/p>\n

8:30<\/strong><\/p>\n

Registrazione Partecipanti<\/em><\/strong><\/p>\n

9:00<\/strong><\/p>\n

Apertura dei Lavori Saluto delle Autorit\u00e0<\/strong><\/p>\n

\u00a0<\/em><\/strong><\/p>\n

I Sessione: <\/em><\/strong>Metodi Computazionali in Chimica Farmaceutica<\/strong><\/em><\/p>\n

\u00a0<\/strong><\/p>\n

9:30<\/strong><\/p>\n

Prof. Vincenzo Barone: \u201c<\/strong>Il ruolo della teoria nelle scienze molecolari\u201d<\/p>\n

10:05<\/strong><\/p>\n

Dott. Matteo Floris: \u201cMMsINC: an alternative chemoproteomics amphitheater\u201d<\/p>\n

10:20<\/strong><\/p>\n

Dott.ssa Lucia Parrotta: \u201cMolecular modeling of DNA G-quadruplex binders\u201d<\/p>\n

10:35<\/strong><\/p>\n

Dott.ssa Marta Del Cadia: \u201cComputational analysis of ligand recognition sites of homo-and heteropentameric 5-HT3 <\/sub>receptors\u201d<\/p>\n

\u00a0<\/p>\n

10:50<\/strong><\/p>\n

Coffee break\/ Poster exhibition<\/strong><\/p>\n

\u00a0<\/p>\n

II Sessione<\/em><\/strong>: Farmaci attivi sul SNC<\/em><\/p>\n

\u00a0<\/em><\/p>\n

11:05<\/strong><\/p>\n

Prof. Gaetano Di Chiara: <\/strong>\u201cPrincipi farmacologici per lo sviluppo di antipsicotici atipici\u201d<\/p>\n

11:40<\/strong><\/p>\n

Dott.ssa Angela De Simone: \u201cA multi-approach study for bace-1 inhibitors characterization\u201d<\/p>\n

11:55<\/strong><\/p>\n

Dott.ssa Francesca Rossi: \u201cSynthesis, biological activity and molecular modeling studies of chalcones and flavones as potential monomine oxidase inhibitors\u00a0\u201d<\/p>\n

12:10<\/strong><\/p>\n

Dott. Gian Cesare Tron: \u201cDiscovery of a nanomolar inhibitor of NMPRTase by click chemistry\u201d<\/p>\n

12:25<\/strong><\/p>\n

Dott.ssa Isabella Pugliesi: \u201cNovel 3-aryl-(1,2,4)triazino(4,3-a)benzimidazol-4(10H)-ones(ATBIs) as selective A2A <\/sub>adenosine receptor antagonists with neuroprotective effect\u201d<\/p>\n

12:40<\/strong><\/p>\n

Dott. Claudio Battilocchio: \u201c1,5-diaryl-pyrroles as new generation of anti-inflammatory and analgesic agents: design, synthesis, in vitro and in vivo evaluation\u201d<\/p>\n

12:55<\/p>\n

Dott.ssa Marina Sala: \u201cStructure-activity relationship of CaMKIINtide peptide analogs<\/p>\n

13:10<\/strong><\/p>\n

Dott.ssa Barbara Parrino: \u201cAnnelated azaindoles with antitumor activity\u201d<\/p>\n

\u00a0<\/p>\n

13:30<\/strong><\/p>\n

Colazione di lavoro<\/p>\n

\u00a0<\/p>\n

III Sessione: <\/em><\/strong>Nuovi approcci terapeutici all\u2019infezione da HIV-1<\/em><\/p>\n

\u00a0<\/p>\n

15:00<\/strong><\/p>\n

Prof. Enzo Tramontano: <\/strong>\u201cNew targets in the early phase of HIV-1 replication\u201d<\/p>\n

15:35<\/strong><\/p>\n

Dott. Valerio Gatti: \u201cIndolylarylsulfones bearing natural and unnatural amino acids as inhibitors of HIV-1 reverse transcriptase and coxsackie B4 virus\u201d<\/p>\n

15:50<\/strong><\/p>\n

Dott. Giosu\u00e8 Costa: \u201cComputational analysis of HIV-1 reverse transcriptase complex\u201d<\/p>\n

16:05<\/strong><\/p>\n

Dott.ssa Irene Briguglio: \u201c(1,2,3)-triazolo-(4,5H)-quinolones. A new class of potent antitubercular agents against multidrug resistant Mycobacterium tuberculosis strains\u201d<\/p>\n

\u00a0<\/p>\n

16:20<\/strong><\/p>\n

Coffee Break\/ Poster exhibition<\/strong><\/p>\n

\u00a0<\/p>\n

IV Sessione: <\/em><\/strong>Nuovi Targets in Chimica Farmaceutica<\/em><\/p>\n

Nuovi Farmaci Antitumorali<\/em><\/p>\n

\u00a0<\/em><\/p>\n

16:35<\/strong><\/p>\n

Prof. Claudia Martini: \u201c<\/strong>Il mitocondrio nel controllo vita\/morte della cellula”<\/p>\n

17:10<\/strong><\/p>\n

Prof. Manlio Palumbo: <\/strong>\u201cNuovi farmaci antitumorali: luci e ombre\u201d<\/em><\/p>\n

17:45<\/strong><\/p>\n

Dott.ssa Maria Tardugno: \u201cBiochemical, Structural, and Biological Evaluation of Tranylcypromine Derivatives as Inhibitors of Histone Demethylases LSD1 and LSD2\u201d<\/p>\n

18:00<\/strong><\/p>\n

Dott.ssa Stefania Sartini: \u201cOne-drug multi target activity. Pyrazolopyrimidine derivatives as antioxidant aldose reductase inhibitors\u201d<\/strong><\/p>\n

18:15<\/strong><\/p>\n

Dott. Giovanni Marzaro: \u201cPsoralenquinone proteasome inhibitors: design, synthesis and biological evaluation\u201d<\/strong><\/p>\n

18:30<\/strong><\/p>\n

Dott. Andrea De Cupertinis: \u201cNew non steroidal agonists of estrogen receptor \u03b2\u201d<\/strong><\/p>\n

18:45<\/strong><\/p>\n

Dott.ssa Sara Bendinelli: \u201cInhibition of mettalloproteinases derived from tumours: new insights in the treatment of human glioblastoma\u201d<\/strong><\/p>\n

19:00<\/strong><\/p>\n

Dott. Antimo Gioiello: \u201cNew Potent and Selective FXR Agonists: Design, Synthesis and Modeling of Norcholanylamine Derivatives\u201d<\/strong><\/p>\n

19:15<\/strong><\/p>\n

Dott.ssa Tracey Pirali: \u201cExploting the reactivity of \u03b1-isocyanoacetamides in diversity-oriented synthesis: an easy access to \u03b1-ketoamides and polysubstituted furans\u201d<\/p>\n

19:30<\/strong><\/p>\n

Dott. Marco Radi: \u201cPlaying around with the decoration of the pyrimidine scaffold: from Non-Nucleoside to Nucleotide-Competing RT Inhibitors\u201d<\/p>\n

\u00a0<\/p>\n

20:30<\/strong><\/p>\n

Cena Sarda<\/p>\n

\u00a0<\/strong><\/p>\n

Venerd\u00ec 07\/05\/2010<\/span><\/strong><\/p>\n

\u00a0<\/strong><\/p>\n

09:00<\/strong><\/p>\n

\u00a0<\/strong><\/p>\n

Prof. Giuseppe Ronsisvalle: <\/strong>\u201cLa qualit\u00e0 nella formazione dottorale e le reti europee\u201d<\/strong><\/p>\n

\u00a0<\/strong><\/p>\n

V Sessione: <\/em><\/strong>\u00a0<\/strong>Metodologie innovative nel Drug Discovery<\/em><\/p>\n

\u00a0<\/strong><\/p>\n

09:20<\/strong><\/p>\n

Dott.ssa Luciana Marinelli:<\/strong><\/p>\n

09:55<\/strong><\/p>\n

Dott.ssa Maria Rosa Buemi: \u201cIdentification of indole derivatives as potent NR2B\/NMDA receptor ligands\u201d<\/strong><\/p>\n

10:10<\/strong><\/p>\n

Dott. Marco Tutone: \u201cInside c-kit tyrosine kinase: molecular modeling and QSAR in the search of new inhibitors\u201d <\/strong><\/p>\n

10:25<\/strong><\/p>\n

Dott. Giovanni Bottegoni: \u201cMultiple receptor conformations enhance early recognition in virtual ligand screening\u201d<\/strong><\/p>\n

\u00a0<\/p>\n

10:40<\/strong><\/p>\n

Coffee Break\/ Poster exhibition<\/p>\n

\u00a0<\/p>\n

\u00a0<\/p>\n

\u00a0<\/p>\n

VI Sessione: <\/em><\/strong>Tecnologie analitiche innovative nel Drug Discovery<\/strong><\/em><\/p>\n

\u00a0<\/p>\n

10:55<\/strong><\/p>\n

Prof.ssa Gabriella Massolini: \u201c<\/strong><\/p>\n

\u00a0<\/strong><\/p>\n

11:30<\/strong><\/p>\n

Dott. Roccaldo Sardella: \u201cDescriptive structure-separation relationship studies in the enantioseparation of amino acids\u201d<\/strong><\/p>\n

11:45<\/strong><\/p>\n

Dott. Marco Pistolozzi: \u201cHPALC and circular dichroism investigation of the tocainide analogues to human serum albumin\u201d<\/strong><\/p>\n

12:00<\/strong><\/p>\n

Dott.ssa Sara Del Carlo: \u201cFluorimetric HPLC analysis of Valdecoxib and Parecoxib: preliminary data\u201d<\/strong><\/p>\n

12:15<\/strong><\/p>\n

Dott.ssa Alessia Bertamino: \u201c<\/strong>Synthesis of Novel Polycyclic Systems by Acid-Catalysed Condensation from a-Amino Aldehydes and L-aminoacids\u201d<\/strong><\/p>\n

12:30<\/strong><\/p>\n

Dott.ssa Valentina Scanzani: \u201cSviluppo e validazione di un metodo in UHPLC di un prodotto farmaceutico\u201d<\/p>\n

\u00a0<\/strong><\/p>\n

12:45<\/strong><\/p>\n

Chiusura dei lavori<\/em><\/p>\n

\u00a0<\/strong><\/p>\n

13:15<\/strong><\/p>\n

Colazione di lavoro<\/strong><\/p>\n","protected":false},"excerpt":{"rendered":"

\u00a0IV Meeting \u201cNuove Prospettive in Chimica Farmaceutica\u201d \u00a0 Gioved\u00ec 06\/05\/2010 8:30 Registrazione Partecipanti 9:00 Apertura dei Lavori Saluto delle Autorit\u00e0 \u00a0 I Sessione: Metodi Computazionali in Chimica Farmaceutica \u00a0 9:30 Prof. Vincenzo Barone: \u201cIl ruolo della teoria nelle scienze molecolari\u201d 10:05 Dott. Matteo Floris: \u201cMMsINC: an alternative chemoproteomics amphitheater\u201d 10:20 Dott.ssa Lucia Parrotta: \u201cMolecular modeling of DNA G-quadruplex binders\u201d 10:35 Dott.ssa Marta Del Cadia: \u201cComputational analysis of ligand recognition sites of homo-and heteropentameric 5-HT3 receptors\u201d \u00a0 10:50 Coffee break\/ Poster exhibition \u00a0 II Sessione: Farmaci attivi sul SNC \u00a0 11:05 Prof. Gaetano Di Chiara: \u201cPrincipi farmacologici per lo sviluppo di […]<\/a><\/p>\n","protected":false},"author":304,"featured_media":0,"parent":65,"menu_order":4,"comment_status":"closed","ping_status":"closed","template":"","meta":{"footnotes":""},"class_list":["post-45","page","type-page","status-publish","hentry","category-918-id","post-seq-1","post-parity-odd","meta-position-corners","fix"],"_links":{"self":[{"href":"https:\/\/people.unica.it\/ivconvegnonpcf\/wp-json\/wp\/v2\/pages\/45","targetHints":{"allow":["GET"]}}],"collection":[{"href":"https:\/\/people.unica.it\/ivconvegnonpcf\/wp-json\/wp\/v2\/pages"}],"about":[{"href":"https:\/\/people.unica.it\/ivconvegnonpcf\/wp-json\/wp\/v2\/types\/page"}],"author":[{"embeddable":true,"href":"https:\/\/people.unica.it\/ivconvegnonpcf\/wp-json\/wp\/v2\/users\/304"}],"replies":[{"embeddable":true,"href":"https:\/\/people.unica.it\/ivconvegnonpcf\/wp-json\/wp\/v2\/comments?post=45"}],"version-history":[{"count":10,"href":"https:\/\/people.unica.it\/ivconvegnonpcf\/wp-json\/wp\/v2\/pages\/45\/revisions"}],"predecessor-version":[{"id":195,"href":"https:\/\/people.unica.it\/ivconvegnonpcf\/wp-json\/wp\/v2\/pages\/45\/revisions\/195"}],"up":[{"embeddable":true,"href":"https:\/\/people.unica.it\/ivconvegnonpcf\/wp-json\/wp\/v2\/pages\/65"}],"wp:attachment":[{"href":"https:\/\/people.unica.it\/ivconvegnonpcf\/wp-json\/wp\/v2\/media?parent=45"}],"curies":[{"name":"wp","href":"https:\/\/api.w.org\/{rel}","templated":true}]}}