| Titolo | Data di pubblicazione | Autori | Tipo | Abstract |
|---|
| Coumarins from Magydaris pastinacea as inhibitors of the tumour-associated carbonic anhydrases IX and XII: isolation, biological studies and in silico evaluation | 2020 | FOIS, BENEDETTA ; DISTINTO, SIMONA ; MELEDDU, RITA ; DEPLANO, SERENELLA ; MACCIONI, ELIAS ; FLORIS, COSTANTINO ; ROSA, ANTONELLA ; NIEDDU, MARIELLA ; CABONI, PIERLUIGI ; Sissi C.; Angeli A.; Supuran C. T.; COTTIGLIA, FILIPPO | 1 Contributo su Rivista::1.1 Articolo in rivista | |
| Investigating the Anticancer Activity of Isatin/Dihydropyrazole Hybrids | 2019 | MELEDDU, RITA ; Petrikaite, Vilma; DISTINTO, SIMONA ; ARRIDU, ANTONELLA ; Angius, Rossella; SERUSI, LORENZO ; Škarnulytė, Laura; Endriulaitytė, Ugnė; Paškevičiu̅tė, Miglė; COTTIGLIA, FILIPPO ; Gaspari, Marco; Taverna, Domenico; DEPLANO, SERENELLA ; FOIS, BENEDETTA ; MACCIONI, ELIAS | 1 Contributo su Rivista::1.1 Articolo in rivista | |
| Novel natural non-nucleoside inhibitors of HIV-1 reverse transcriptase identified by shape- and structure-based virtual screening techniques | 2019 | Giosuè Costa; Roberta Rocca; CORONA, ANGELA ; GRANDI, NICOLE ; Federica Moraca; Isabella Romeo; Carmine Talarico; Maria Giovanna Gagliardi; Francesca Alessandra Ambrosio; Francesco Ortuso; Stefano Alcaro; DISTINTO, SIMONA ; MACCIONI, ELIAS ; TRAMONTANO, ENZO ; Anna Artese | 1 Contributo su Rivista::1.1 Articolo in rivista | |
| From cycloheptathiophene-3-carboxamide to oxazinone-based derivatives as allosteric HIV-1 ribonuclease H inhibitors | 2019 | Serena Massari; CORONA, ANGELA ; DISTINTO, SIMONA ; Jenny Desantis; CAREDDA, ALESSIA ; Stefano Sabatini; Giuseppe Manfroni; Tommaso Felicetti; Violetta Cecchetti; Christophe Pannecouque; MACCIONI, ELIAS ; TRAMONTANO, ENZO ; Oriana Tabarrini | 1 Contributo su Rivista::1.1 Articolo in rivista | |
| Ferulic Acid Esters and Withanolides: in Search of Withania somnifera GABAA Receptor Modulators | 2019 | SONAR, VIJAY PRAKASH ; FOIS, BENEDETTA ; DISTINTO, SIMONA ; MACCIONI, ELIAS ; MELEDDU, RITA ; COTTIGLIA, FILIPPO ; ACQUAS, ELIO MARIA GIOACHINO ; Sanjay Kasture; FLORIS, COSTANTINO ; Daniele Colombo; SISSI, CLAUDIA ; SANNA, ENRICO ; TALANI, GIUSEPPE | 1 Contributo su Rivista::1.1 Articolo in rivista | |
| Exploring new structural features of the 4-[(3-methyl-4-aryl-2,3-dihydro-1,3-thiazol-2-ylidene)amino]benzenesulphonamide scaffold for the inhibition of human carbonic anhydrases | 2019 | DISTINTO, SIMONA ; MELEDDU, RITA ; Ortuso F.; COTTIGLIA, FILIPPO ; DEPLANO, SERENELLA ; SOUSA SEQUEIRA, ANA LISA ; MELIS, CLAUDIA ; FOIS, BENEDETTA ; Angeli A.; Capasso C.; ANGIUS, RICCARDO ; Alcaro S.; Supuran C. T.; MACCIONI, ELIAS | 1 Contributo su Rivista::1.1 Articolo in rivista | |
| Targeting tumor associated carbonic anhydrase IX and XII: Highly isozyme selective coumarin and psoralen inhibitors | 2018 | MELIS, CLAUDIA ; DISTINTO, SIMONA ; BIANCO, GIULIA ; MELEDDU, RITA ; COTTIGLIA, FILIPPO ; FOIS, BENEDETTA ; Taverna, Domenico; Angius, Rossella; Alcaro, Stefano; Ortuso, Francesco; Gaspari, Marco; Angeli, Andrea; Del Prete, Sonia; Capasso, Clemente; Supuran, Claudiu T.; MACCIONI, ELIAS | 1 Contributo su Rivista::1.1 Articolo in rivista | |
| Identification of Myricetin as Ebolavirus VP35-dsRNA interaction inhibitor through a novel fluorescence-based assay | 2018 | Gian Luca Daino; FRAU, ALDO ; SANNA, CINZIA ; Daniela Rigano; DISTINTO, SIMONA ; MADAU, VERONICA ; ESPOSITO, FRANCESCA ; FANUNZA, ELISA ; BIANCO, GIULIA ; Orazio Taglialatela-Scafati; ZINZULA, LUCA ; MACCIONI, ELIAS ; CORONA, ANGELA ; TRAMONTANO, ENZO | 1 Contributo su Rivista::1.1 Articolo in rivista | |
| Tuning the Dual Inhibition of Carbonic Anhydrase and Cyclooxygenase by Dihydrothiazole Benzensulfonamides | 2018 | MELEDDU, RITA ; DISTINTO, SIMONA ; COTTIGLIA, FILIPPO ; Angius Rossella; Gaspari Marco; Taverna Domenico; MELIS, CLAUDIA ; Angeli Andrea; BIANCO, GIULIA ; DEPLANO, SERENELLA ; FOIS, BENEDETTA ; Del Prete Sonia; Capasso Clemente; Alcaro Stefano; Ortuso Francesco; Yanez Matilde; Supuran Claudiu T.; MACCIONI, ELIAS | 1 Contributo su Rivista::1.1 Articolo in rivista | |
| Phenylpropenoids from Bupleurum fruticosum as Anti-Human Rhinovirus Species A Selective Capsid Binders | 2017 | FOIS, BENEDETTA ; BIANCO, GIULIA ; SONAR, VIJAY PRAKASH ; DISTINTO, SIMONA ; MACCIONI, ELIAS ; MELEDDU, RITA ; Melis, Claudia; MARRAS, LUISA ; POMPEI, RAFFAELLO ; FLORIS, COSTANTINO ; CABONI, PIERLUIGI ; COTTIGLIA, FILIPPO | 1 Contributo su Rivista::1.1 Articolo in rivista | |
| Through scaffold modification to 3,5-diaryl-4,5-dihydroisoxazoles: new potent and selective inhibitors of monoamine oxidase B | 2017 | MELEDDU, RITA ; DISTINTO, SIMONA ; Cirilli, Roberto; Alcaro, Stefano; Yanez, Matilde; SANNA, MARIA LUISA ; CORONA, ANGELA ; MELIS, CLAUDIA ; BIANCO, GIULIA ; Matyus, Peter; COTTIGLIA, FILIPPO ; MACCIONI, ELIAS | 1 Contributo su Rivista::1.1 Articolo in rivista | |
| Design, synthesis and antiviral evaluation of novel heteroarylcarbothioamide derivatives as dual inhibitors of HIV-1 Reverse transcriptase-associated RNase H and RDDP functions | 2017 | CORONA, ANGELA ; ONNIS, VALENTINA ; DEPLANO, ALESSANDRO ; BIANCO, GIULIA ; DEMURTAS, MONICA ; DISTINTO, SIMONA ; Cheng, Yung Chi; Alcaro, Stefano; ESPOSITO, FRANCESCA ; TRAMONTANO, ENZO | 1 Contributo su Rivista::1.1 Articolo in rivista | |
| Natural product-inspired esters and amides of ferulic and caffeic acid as dual inhibitors of HIV-1 reverse transcriptase | 2017 | SONAR, VIJAY PRAKASH ; CORONA, ANGELA ; DISTINTO, SIMONA ; MACCIONI, ELIAS ; MELEDDU, RITA ; FOIS, BENEDETTA ; FLORIS, COSTANTINO ; Malpure, Nilesh V.; Alcaro, Stefano; TRAMONTANO, ENZO ; COTTIGLIA, FILIPPO | 1 Contributo su Rivista::1.1 Articolo in rivista | |
| N-Acylbenzenesulfonamide dihydro-1,3,4-oxadiazole hybrids: seeking selectivity toward carbonic anhydrase isoforms | 2017 | BIANCO, GIULIA ; MELEDDU, RITA ; DISTINTO, SIMONA ; COTTIGLIA, FILIPPO ; Gaspari, Marco; MELIS, CLAUDIA ; CORONA, ANGELA ; Angius, Rossella; Angeli, Andrea; Taverna, Domenico; Alcaro, Stefano; Leitans, Janis; Kazaks, Andris; Tars, Kaspars; Supuran, Claudiu T.; MACCIONI, ELIAS | 1 Contributo su Rivista::1.1 Articolo in rivista | |
| Multi-target activity of Hemidesmus indicus decoction against innovative HIV-1 drug targets and characterization of Lupeol mode of action | 2017 | ESPOSITO, FRANCESCA ; Mandrone, Manuela; Del Vecchio, Claudia; Carli, Ilaria; DISTINTO, SIMONA ; CORONA, ANGELA ; Lianza, Mariacaterina; PIANO, DARIO ; Tacchini, Massimo; MACCIONI, ELIAS ; COTTIGLIA, FILIPPO ; Saccon, Elisa; Poli, Ferruccio; Parolin, Cristina; TRAMONTANO, ENZO | 1 Contributo su Rivista::1.1 Articolo in rivista | |
| Isatin: a privileged scaffold for the design of carbonic anhydrase inhibitors | 2017 | MELIS, CLAUDIA ; MELEDDU, RITA ; Angeli, Andrea; DISTINTO, SIMONA ; BIANCO, GIULIA ; Capasso, Clemente; COTTIGLIA, FILIPPO ; Angius, Rossella; Supuran, Claudiu T.; MACCIONI, ELIAS | 1 Contributo su Rivista::1.1 Articolo in rivista | |
| Isatin thiazoline hybrids as dual inhibitors of HIV-1 reverse transcriptase | 2017 | MELEDDU, RITA ; DISTINTO, SIMONA ; CORONA, ANGELA ; TRAMONTANO, ENZO ; BIANCO, GIULIA ; MELIS, CLAUDIA ; COTTIGLIA, FILIPPO ; MACCIONI, ELIAS | 1 Contributo su Rivista::1.1 Articolo in rivista | |
| Drug design, synthesis, in vitro and in silico evaluation of selective monoaminoxidase B inhibitors based on 3-acetyl-2-dichlorophenyl-5-aryl-2,3-dihydro-1,3,4-oxadiazole chemical scaffold | 2016 | DISTINTO, SIMONA ; MELEDDU, RITA ; Yanez, Matilde; Cirilli, Roberto; BIANCO, GIULIA ; SANNA, MARIA LUISA ; ARRIDU, ANTONELLA ; Cossu, Pietro; COTTIGLIA, FILIPPO ; Faggi, Cristina; Ortuso, Francesco; Alcaro, Stefano; MACCIONI, ELIAS | 1 Contributo su Rivista::1.1 Articolo in rivista | |
| Sennoside A, derived from the traditional chinese medicine plant Rheum L., is a new dual HIV-1 inhibitor effective on HIV-1 replication | 2016 | ESPOSITO, FRANCESCA ; Carli, Ilaria; Del Vecchio, Claudia; Xu, Lijia; CORONA, ANGELA ; GRANDI, NICOLE ; PIANO, DARIO ; MACCIONI, ELIAS ; DISTINTO, SIMONA ; Parolin, Cristina; TRAMONTANO, ENZO | 1 Contributo su Rivista::1.1 Articolo in rivista | |
| Studies on Cycloheptathiophene-3-carboxamide Derivatives as Allosteric HIV-1 Ribonuclease H Inhibitors | 2016 | CORONA, ANGELA ; Desantis, Jenny; Massari, Serena; DISTINTO, SIMONA ; Masaoka, Takashi; Sabatini, Stefano; ESPOSITO, FRANCESCA ; Manfroni, Giuseppe; MACCIONI, ELIAS ; Cecchetti, Violetta; Pannecouque, Christophe; Le Grice, Stuart F. J; TRAMONTANO, ENZO ; Tabarrini, Oriana | 1 Contributo su Rivista::1.1 Articolo in rivista | |
