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TitoloData di pubblicazioneAutore(i)RivistaEditore
Sulfonamide/sulfamate switch with a series of piperazinylureido derivatives: Synthesis, kinetic and in silico evaluation as carbonic anhydrase isoforms I, II, IV, and IX inhibitors2020Nocentini, Alessio; Moi, Davide; Deplano, Alessandro; Osman, Sameh M.; AlOthman, Zeid A.; Balboni..., Gianfranco; Supuran, Claudiu T.; Onnis, ValentinaEUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
Appliance of the piperidinyl-hydrazidoureido linker to benzenesulfonamide compounds: Synthesis, in vitro and in silico evaluation of potent carbonic anhydrase II, IX and XII inhibitors2020Moi, Davide; Nocentini, Alessio; Deplano, Alessandro; Osman, Sameh M.; AlOthman, Zeid A.; Piras, ...Valentina; Balboni, Gianfranco; Supuran, Claudiu T.; Onnis, ValentinaBIOORGANIC CHEMISTRY
Exploring the fatty acid amide hydrolase and cyclooxygenase inhibitory properties of novel amide derivatives of ibuprofen2020Deplano, Alessandro; Karlsson, Jessica; Svensson, Mona; Moraca, Federica; Catalanotti, Bruno; Fow...ler, Christopher J.; Onnis, ValentinaJOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
The fatty acid amide hydrolase and cyclooxygenase-inhibitory properties of novel amide derivatives of carprofen2020Deplano, Alessandro; Karlsson, Jessica; Fowler, Christopher J.; Onnis, ValentinaBIOORGANIC CHEMISTRY
Benzylamides and piperazinoarylamides of ibuprofen as fatty acid amide hydrolase inhibitors2019Deplano, Alessandro; Cipriano, Mariateresa; Moraca, Federica; Novellino, Ettore; Catalanotti, Bru...no; Fowler, Christopher J.; Onnis, ValentinaJOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
Structure-activity relationship with pyrazoline-based aromatic sulfamates as carbonic anhydrase isoforms I, II, IX and XII inhibitors: Synthesis and biological evaluation2019Moi, Davide; Nocentini, Alessio; Deplano, Alessandro; Balboni, Gianfranco; Supuran, Claudiu T.; O...nnis, ValentinaEUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
Synthesis and in vitro evaluation of piperazinyl-ureido sulfamates as steroid sulfatase inhibitors2019Moi, Davide; Foster, Paul A.; Rimmer, Lucy G.; Jaffri, Alisha; Deplano, Alessandro; Balboni, Gian...franco; Onnis, Valentina; Potter, Barry V. L.EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
Hydrophobic similarity between molecules: Application to three-dimensional molecular overlays with PharmScreen2018Vazquez, Javier; Deplano, Alessandro; Herrero, Albert; Gibert, Enric; Ginex, Tiziana; Rabal, Obdu...lia; Oyarzabal, Julen; Herrero, Enric; Luque, F JavierAmerican Chemical Society
Development and Validation of Molecular Overlays Derived from Three-Dimensional Hydrophobic Similarity with PharmScreen2018Vázquez, J.; Deplano, A.; Herrero, A.; Ginex, T.; Gibert, E.; Rabal, O.; Oyarzabal, J.; Herrero, ...E.; Luque, F. J.JOURNAL OF CHEMICAL INFORMATION AND MODELING
Onthe use (QM) IEF/PMC-MST-derived hydrophobic contributions as physicochemical descriptors in 3D-QSAR: the PHARMSQSARTM approach2018Rey, Oscar; Ginex, Tiziana; Vazquez, Javier; Deplano, Alessandro; Herrero, Albert; Gibert, Enric;... Herrero, Enric; Javier Luque, Francisco
Novel propanamides as fatty acid amide hydrolase inhibitors2017Deplano, Alessandro; Morgillo, Carmine Marco; Demurtas, Monica; Björklund, Emmelie; Cipriano, Mar...iateresa; Svensson, Mona; Hashemian, Sanaz; Smaldone, Giovanni; Pedone, Emilia; Luque, F. Javier; Cabiddu, MARIA GRAZIA; Novellino, Ettore; Fowler, Christopher J.; Catalanotti, Bruno; Onnis, ValentinaEUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
Design, synthesis and antiviral evaluation of novel heteroarylcarbothioamide derivatives as dual inhibitors of HIV-1 Reverse transcriptase-associated RNase H and RDDP functions2017Corona, Angela; Onnis, Valentina; Deplano, Alessandro; Bianco, Giulia; Demurtas, Monica; Distinto..., Simona; Cheng, Yung Chi; Alcaro, Stefano; Esposito, Francesca; Tramontano, EnzoPATHOGENS AND DISEASE
Design, synthesis and SAR of small molecules acting on pain pathways24-mar-2016Università degli Studi di Cagliari
DIHYDROQUINAZOLINE BENZYLAMIDES AS ACETYLCHOLINESTERASE AND BUTYRYLCHOLINESTERASE INHIBITORS2016Onnis, Valentina; Balboni, Gianfranco; Deplano, Alessandro; Demurtas, Monica; Buyn, Joon Seok; So...hn, Joo Mi; Lee, Jae Yeol; Catto, Marco; Pisani, Leonardo; Carotti, Angelo
Potent nematicidal activity of maleimide derivatives on Meloidogyne incognita2016Eloh, K; Demurtas, M; Mura, MG; Deplano, A; Onnis, V; Sasanelli, N; Maxia, A; Caboni, PJOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY
Design, synthesis and evaluation of antiproliferative activity of new benzimidazolehydrazones2016Onnis, V; Demurtas, M; Deplano, A; Balboni, G; Baldisserotto, A; Manfredini, S; Pacifico, S; Liek...ens, S; Balzarini, JMOLECULES
Discovery of a novel class of profen derivatives as FAAH inhibitors: MD and QM/MM studies of the binding mode and 3D SAR2016Morgillo, CM; Deplano, A; Karlsson, J; Cipriano, M; Björklund, E; Fowler, Cj; Onnis, V; Luque, Fj...; Catalanotti, B
DESIGN, SYNTHESIS AND PHARMACOLOGICAL INVESTIGATION OF NEW DNA METHYLTRANSFERASE INHIBITORS2016Balboni, Gianfranco; Deplano, Alessandro; Demurtas, Monica; Arimondo, Paola B.; Masson, Veronique...; Onnis, Valentina
Homology modeling of a Class A GPCR in the inactive conformation: A quantitative analysis of the correlation between model/template sequence identity and model accuracy2016Costanzi, Stefano; Skorski, Matthew; Deplano, Alessandro; Habermehl, Brett; Mendoza, Mary; Wang, ...Keyun; Biederman, Michelle; Dawson, Jessica; Gaoa, JiaJOURNAL OF MOLECULAR GRAPHICS & MODELLING
Inhibitory effect of positively charged triazine antagonists of prokinecitin receptors on the transient receptor vanilloid type-1 (TRPV1) channel2015Petrocellis, Luciano De; Moriello, Aniello Schiano; Byun, Joon Seok; Sohn, Joo Mi; Lee, Jae Yeol;... Vázquez-Romero, Ana; Garrido, Maria; Messeguer, Angel; Zhang, Fang-Xiong; Zamponi, Gerald W; Deplano, Alessandro; Congiu, Cenzo; Onnis, Valentina; Balboni, Gianfranco; Marzo, Vincenzo DiPHARMACOLOGICAL RESEARCH
   
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