Prodotti della ricerca
UNICA IRIS Institutional Research Information System
IRIS è il sistema di gestione integrata dei dati della ricerca (persone, progetti, pubblicazioni, attività) adottato dall'Università degli Studi di Cagliari dal mese di luglio 2015.

Titolo | Data di pubblicazione | Autore(i) | Rivista | Editore |
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Synthesis and evaluation of antioxidant and antiproliferative activity of 2-arylbenzimidazoles | 2020 | Baldisserotto, Anna; Demurtas, Monica; Lampronti, Ilaria; Tacchini, Massimo; Moi, Davide; Balboni..., Gianfranco; Pacifico, Salvatore; Vertuani, Silvia; Manfredini, Stefano; Onnis, Valentina | BIOORGANIC CHEMISTRY | |
Appliance of the piperidinyl-hydrazidoureido linker to benzenesulfonamide compounds: Synthesis, in vitro and in silico evaluation of potent carbonic anhydrase II, IX and XII inhibitors | 2020 | Moi, Davide; Nocentini, Alessio; Deplano, Alessandro; Osman, Sameh M.; AlOthman, Zeid A.; Piras, ...Valentina; Balboni, Gianfranco; Supuran, Claudiu T.; Onnis, Valentina | BIOORGANIC CHEMISTRY | |
The fatty acid amide hydrolase and cyclooxygenase-inhibitory properties of novel amide derivatives of carprofen | 2020 | Deplano, Alessandro; Karlsson, Jessica; Fowler, Christopher J.; Onnis, Valentina | BIOORGANIC CHEMISTRY | |
Sulfonamide/sulfamate switch with a series of piperazinylureido derivatives: Synthesis, kinetic and in silico evaluation as carbonic anhydrase isoforms I, II, IV, and IX inhibitors | 2020 | Nocentini, Alessio; Moi, Davide; Deplano, Alessandro; Osman, Sameh M.; AlOthman, Zeid A.; Balboni..., Gianfranco; Supuran, Claudiu T.; Onnis, Valentina | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | |
Ruthenium(II) Complexes of Isothiazole Ligands: Crystal Structure, HSA/DNA Interactions, Cytotoxic Activity and Molecular Docking Simulations | 2020 | Djukić, Maja B.; Jeremić, Marija S.; Filipović, Ignjat P.; Klisurić, Olivera R.; Jelić, Ratomir M....; Popović, Suzana; Matić, Sanja; Onnis, Valentina; Matović, Zoran D. | CHEMISTRYSELECT | |
2-(Arylamino)-6-(trifluoromethyl)nicotinic Acid Derivatives: New HIV-1 RT Dual Inhibitors Active on Viral Replication | 2020 | Corona, Angela; Onnis, Valentina; Del Vecchio, Claudia; Esposito, Francesca; Cheng, Yung-Chi; Tra...montano, Enzo | MOLECULES | |
Synthesis and Biological Evaluation of 2-Substituted Benzyl-/Phenylethylamino-4-amino-5-aroylthiazoles as Apoptosis-Inducing Anticancer Agents | 2020 | Oliva, Paola; Onnis, Valentina; Balboni, Elisa; Hamel, Ernest; Estévez-Sarmiento, Francisco; Quin...tana, José; Estévez, Francisco; Brancale, Andrea; Ferla, Salvatore; Manfredini, Stefano; Romagnoli, Romeo | MOLECULES | |
Exploring the fatty acid amide hydrolase and cyclooxygenase inhibitory properties of novel amide derivatives of ibuprofen | 2020 | Deplano, Alessandro; Karlsson, Jessica; Svensson, Mona; Moraca, Federica; Catalanotti, Bruno; Fow...ler, Christopher J.; Onnis, Valentina | JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY | |
Response to Perspectives on the Classical Enzyme Carbonic Anhydrase and the Search for Inhibitors | 2020 | Angeli, Andrea; Carta, Fabrizio; Nocentini, Alessio; Winum, Jean-Yves; Zalubovskis, Raivis; Onnis..., Valentina; Eldehna, Wagdy M; Capasso, Clemente; Carradori, Simone; Donald, William A; Dedhar, Shoukat; Supuran, Claudiu T | BIOPHYSICAL JOURNAL | |
In-Vitro Evaluation of Antioxidant, Antiproliferative and Photo-Protective Activities of Benzimidazolehydrazone Derivatives | 2020 | Baldisserotto, Anna; Demurtas, Monica; Lampronti, Ilaria; Tacchini, Massimo; Moi, Davide; Balboni..., Gianfranco; Vertuani, Silvia; Manfredini, Stefano; Onnis, Valentina | PHARMACEUTICALS | |
Carbonic anhydrase inhibitors targeting metabolism and tumor microenvironment | 2020 | Angeli, Andrea; Carta, Fabrizio; Nocentini, Alessio; Winum, Jean-Yves; Zalubovskis, Raivis; Akdem...ir, Atilla; Onnis, Valentina; Eldehna, Wagdy M.; Capasso, Clemente; Simone, Giuseppina De; Monti, Simona Maria; Carradori, Simone; Donald, William A.; Dedhar, Shoukat; Supuran, Claudiu T. | METABOLITES | |
Indole derivatives as multifunctional drugs: Synthesis and evaluation of antioxidant, photoprotective and antiproliferative activity of indole hydrazones | 2019 | Demurtas, Monica; Baldisserotto, Anna; Lampronti, Ilaria; Moi, Davide; Balboni, Gianfranco; Pacif...ico, Salvatore; Vertuani, Silvia; Manfredini, Stefano; Onnis, Valentina | BIOORGANIC CHEMISTRY | |
Synthesis and in vitro evaluation of piperazinyl-ureido sulfamates as steroid sulfatase inhibitors | 2019 | Moi, Davide; Foster, Paul A.; Rimmer, Lucy G.; Jaffri, Alisha; Deplano, Alessandro; Balboni, Gian...franco; Onnis, Valentina; Potter, Barry V. L. | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | |
Structure-activity relationship with pyrazoline-based aromatic sulfamates as carbonic anhydrase isoforms I, II, IX and XII inhibitors: Synthesis and biological evaluation | 2019 | Moi, Davide; Nocentini, Alessio; Deplano, Alessandro; Balboni, Gianfranco; Supuran, Claudiu T.; O...nnis, Valentina | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | |
Benzylamides and piperazinoarylamides of ibuprofen as fatty acid amide hydrolase inhibitors | 2019 | Deplano, Alessandro; Cipriano, Mariateresa; Moraca, Federica; Novellino, Ettore; Catalanotti, Bru...no; Fowler, Christopher J.; Onnis, Valentina | JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY | |
Targeting prokineticin system counteracts hypersensitivity, neuroinflammation, and tissue damage in a mouse model of bortezomib-induced peripheral neuropathy | 2019 | Moschetti, Giorgia; Amodeo, Giada; Maftei, Daniela; Lattanzi, Roberta; Procacci, Patrizia; Sartor...i, Patrizia; Balboni, Gianfranco; Onnis, Valentina; Conte, Vincenzo; Panerai, Alberto; Sacerdote, Paola; Franchi, Silvia | JOURNAL OF NEUROINFLAMMATION | |
Discovery of thiazolin-4-one-based aromatic sulfamates as a new class of carbonic anhydrase isoforms I, II, IV, and IX inhibitors | 2018 | Nocentini, Alessio; Moi, Davide; Balboni, Gianfranco; Onnis, Valentina; Supuran, Claudiu T. | BIOORGANIC CHEMISTRY | |
Benzofuran hydrazones as potential scaffold in the development of multifunctional drugs: Synthesis and evaluation of antioxidant, photoprotective and antiproliferative activity | 2018 | Baldisserotto, Anna; Demurtas, Monica; Lampronti, Ilaria; Moi, Davide; Balboni, Gianfranco; Vertu...ani, Silvia; Manfredini, Stefano; Onnis, Valentina | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY | |
Synthesis and biological evaluation of novel pyrazoline-based aromatic sulfamates with potent carbonic anhydrase isoforms II, IV and IX inhibitory efficacy | 2018 | Nocentini, Alessio; Moi, Davide; Balboni, Gianfranco; Salvadori, Severo; Onnis, Valentina; Supura...n, Claudiu T. | BIOORGANIC CHEMISTRY | |
3,4-Dihydroquinazoline derivatives inhibit the activities of cholinesterase enzymes | 2017 | Park, Byeongyeon; Nam, Ji Hye; Kim, Jin Han; Kim, Hyoung Ja; Onnis, Valentina; Balboni, Gianfranc...o; Lee, Kyung Tae; Park, Jeong Ho; Catto, Marco; Carotti, Angelo; Lee, Jae Yeol | BIOORGANIC & MEDICINAL CHEMISTRY LETTERS | Elsevier Ltd |